1206161-97-8
- Product Name：Filgotinib
- Molecular Formula：
- Purity：99%
- Molecular Weight：425.511
Product Details;
CasNo： 1206161-97-8
Buy cost-effective 99% pure Filgotinib 1206161-97-8 now
- Molecular Formula:C21H23N5O3S
- Molecular Weight:425.511
- PKA:8.04±0.20(Predicted)
- Density:1.51±0.1 g/cm3(Predicted)
1206161-97-8 Relevant articles
PROCESSES FOR THE PREPARATION OF FILGOTINIB
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Paragraph 0080-0081, (2020/03/09)
The present invention relates to process...
Preparation method of filgotinib
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Paragraph 0084-0087, (2020/03/23)
A preparation method of filgotinib compr...
NOVEL PROCESS FOR THE PREPARATION OF FILGOTINIB AND INTERMEDIATES THEREOF
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Page/Page column 17-18, (2020/10/20)
The present invention relates to a novel...
Synthesis method of JAK1 inhibitor Filgotinib
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Paragraph 0062-0064; 0073-0077, (2019/10/01)
The invention provides a preparing metho...
1206161-97-8 Process route
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![5-[4-(1,1-dioxothiomorpholin-4-ylmethyl)-phenyl]-[1,2,4]triazolo[1,5-a]pyridin-2-ylamine](/upload/2026/7/88f4eb60-f048-4b44-82e4-549c7790cb22.png)
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1257705-09-1
5-[4-(1,1-dioxothiomorpholin-4-ylmethyl)-phenyl]-[1,2,4]triazolo[1,5-a]pyridin-2-ylamine
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4023-34-1
cyclopropanecarboxylic acid chloride
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1206161-97-8
N-(5-{4-[(1,1-dioxo-1λ6-thiomorpholin-4-yl)methyl]phenyl}-[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamide
| Conditions | Yield |
|---|---|
|
With
4-methyl-morpholine;
In
1,4-dioxane;
at 50 ℃;
for 4h;
Reagent/catalyst;
Solvent;
Temperature;
Green chemistry;
|
91.2% |
|
With
triethylamine;
at 5 - 20 ℃;
|
-
-
C25H27N5O4S
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1206161-97-8
N-(5-{4-[(1,1-dioxo-1λ6-thiomorpholin-4-yl)methyl]phenyl}-[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamide
| Conditions | Yield |
|---|---|
|
With
ammonium hydroxide;
In
ethanol;
at 20 ℃;
Reagent/catalyst;
Solvent;
|
94.3% |
1206161-97-8 Upstream products
-
39093-93-1
thiomorpholine 1,1-dioxide
-
1206163-59-8
cyclopropanecarboxylic acid [5-(4-bromomethyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]-amide
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1142936-49-9
cyclopropanecarboxylic acid [5-(4-hydroxymethyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]-amide
-
19798-81-3
2-Amino-6-bromopyridine
1206161-97-8 Downstream products
-
1257705-09-1
5-[4-(1,1-dioxothiomorpholin-4-ylmethyl)-phenyl]-[1,2,4]triazolo[1,5-a]pyridin-2-ylamine
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